PUBLICATIONS
Covalent Protein Inhibitors via Tyrosine and Tryptophan Conjugation with Cyclic Imine Mannich Electrophiles
Wang, S.*, Wang, L.*, Hadisurya, M., Shahbazi Nia, S., Tao, W. A., Dykhuizen, E. C., Krusemark, C. J., In press at Angewandte Chemie Int. Ed.
Assays of DNA-encoded Libraries Against Protein Targets On and Within Living Cells
Shahbazi Nia, S., Krusemark, C. J., In Liu, G., Krusemark, C. J., Li, J. (Eds.), DNA-encoded Library Technology for Drug Discovery, (2025) 85, 63-86. Royal Society of Chemistry. DOI: 10.1039/9781788016032-00063
Selections of DNA-Encoded Libraries to Protein Targets on Living Cells
Cai, B.., Krusemark, C. J., In Scheuermann, J., Li, Y (Eds.), Science of Synthesis: DNA-Encoded Libraries, (2024) 1, 599. Thieme.
Selections of DNA-Encoded Libraries to Protein Targets within Living Cells
Cai, B.., Krusemark, C. J., In Scheuermann, J., Li, Y (Eds.), Science of Synthesis: DNA-Encoded Libraries, (2024) 1, 607. Thieme.
Direct Selection of DNA-encoded Libraries for Biased Agonists of GPCRs on Live Cells.
Cai, B., El Daibani, A., Bai, Y., Che, T., Krusemark, C. J., JACS Au, 2023, 3, 4, 1076–1088.
“Selection Methods for Proximity-dependent Enrichment of Ligands from DNA-encoded Chemical Libraries using Enzymatic Fusion Proteins.
Cai, B., Mhetre, A. B., Krusemark, C. J., Chemical Science. 2023, 14, 245-250.
Covalent Protein Inhibitors via Tyrosine Conjugation with Cyclic Imine Mannich Electrophiles.
Wang, S., Hadisurya, M., Tao, W. A., Dykhuizen, E. C., Krusemark, C. J., ChemRxiv. 2022
Multiplexed Small Molecule Ligand Binding Assays by Affinity Labeling and DNA Sequence Analysis
Cai, B., Krusemark, C. J., Angewandte Chemie Int. Ed. 2022, 61, 3, e20213515
Discovery and Characterization of a Potent, Selective, and Cellularly Active CBX2 Chromodomain Ligand
Wang, S., Alpsoy, A., Sood, S., Dhiman, A., Ordonex-Rubiano, S., Sun, Y., Jiao, G., Krusemark, C. J., Dykhuizen, E. C. ChemBioChem 2021, 22, 2335-2344